OBJECTIVE To evaluate the feasibility of LHRH-A2-loaded monostearin solid lipid nanoparticles ( LHRH-A2-MSLN) as a novel preparation for oral administration. 目的考察以固体脂质纳米粒为载体包裹促黄体生成素释放激素的类似物(LHRH-A2)口服给药的可行性。
Lipid ( Monostearin) and surfactant were used to prepare ARE-SLN by heating-ultrasound divergence method and solvent-emulsion method respectively. 对于固体脂质纳米粒的制备,分别进行两种制备方法的研究:热融超声分散法和溶剂乳化法。